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GAK inhibitor 49
CAS No. 319492-82-5
GAK inhibitor 49( —— )
Catalog No. M22093 CAS No. 319492-82-5
GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 178 | In Stock |
|
| 10MG | 295 | In Stock |
|
| 25MG | 498 | In Stock |
|
| 50MG | 716 | In Stock |
|
| 100MG | 981 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameGAK inhibitor 49
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NoteResearch use only, not for human use.
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Brief DescriptionGAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
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DescriptionGAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
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In VitroGAK inhibitor 49 (compound 49) shows a weak inhibitory effect on AAK1, BMP2K and STK16, with IC50s of 28, 63 and >100 μM, respectively.
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorGAK
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Research Area——
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Indication——
Chemical Information
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CAS Number319492-82-5
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Formula Weight370.4
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Molecular FormulaC20H22N2O5?
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (134.99 mM)
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SMILESCOc1cc2nccc(Nc3cc(OC)c(OC)c(OC)c3)c2cc1OC
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Asquith CRM, et al. Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase. ChemMedChem. 2018;13(1):48-66.
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