GAK inhibitor 49

CAS No. 319492-82-5

GAK inhibitor 49 ( —— )

Catalog No. M22093 CAS No. 319492-82-5

GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 178 In Stock
10MG 295 In Stock
25MG 498 In Stock
50MG 716 In Stock
100MG 981 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    GAK inhibitor 49
  • Note
    Research use only, not for human use.
  • Brief Description
    GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
  • Description
    GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GAK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    319492-82-5
  • Formula Weight
    370.4
  • Molecular Formula
    C20H22N2O5?
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    COc1cc2nccc(Nc3cc(OC)c(OC)c(OC)c3)c2cc1OC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Asquith CRM, et al. Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase. ChemMedChem. 2018;13(1):48-66.
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